Title
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Synthesis of 4-aminoquinolines by aerobic oxidative palladium-catalyzed double CH activation and isocyanide insertion
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Author
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Abstract
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An unprecedented aerobic oxidative Pd-catalyzed imidoylative coupling of two CH fragments furnishing medicinally valuable 4-aminoquinolines is reported. Optimization studies are described and several analogs were successfully prepared. |
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Language
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English
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Source (journal)
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Chemistry of heterocyclic compounds. - New York
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Publication
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New York
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2013
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ISSN
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0009-3122
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DOI
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10.1007/S10593-013-1324-Z
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Volume/pages
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49
:6
(2013)
, p. 902-908
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ISI
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000324215000010
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Full text (Publisher's DOI)
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Full text (publisher's version - intranet only)
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