Title
Extending the scope of the Aza-Fischer synthesis of 4- and 6-azaindoles Extending the scope of the Aza-Fischer synthesis of 4- and 6-azaindoles
Author
Faculty/Department
Faculty of Pharmaceutical, Biomedical and Veterinary Sciences. Pharmacy
Publication type
article
Publication
Weinheim ,
Subject
Chemistry
Source (journal)
European journal of organic chemistry. - Weinheim
Volume/pages
(2013) :16 , p. 3328-3336
ISSN
1434-193X
Carrier
E
Target language
English (eng)
Full text (Publishers DOI)
Abstract
Fischer indole cyclization has recently been described as an efficient approach to the synthesis of azaindoles bearing electron-donating groups. We now show that this cascade reaction can be very efficient for the formation of a wider range of 4- and 6-azaindoles by using microwave irradiation.
E-info
https://repository.uantwerpen.be/docman/iruaauth/4dc48b/760d035c3cc.pdf