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Title
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Novel selective glucocorticoid receptor agonists (SEGRAs) with a covalent warhead for long-lasting inhibition
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Author
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Abstract
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| The synthesis and in vitro properties of six analogues of the selective glucocorticoid receptor (GR) agonist GSK866, bearing a warhead for covalent linkage to the glucocorticoid receptor, is described. |
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Language
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English
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Source (journal)
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Bioorganic and medicinal chemistry letters. - Oxford
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Publication
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Oxford
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2016
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ISSN
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0960-894X
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DOI
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10.1016/J.BMCL.2016.08.091
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Volume/pages
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26
:20
(2016)
, p. 5032-5038
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ISI
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000385498500036
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Full text (Publisher's DOI)
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Full text (open access)
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Full text (publisher's version - intranet only)
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