Publication
Title
Novel selective glucocorticoid receptor agonists (SEGRAs) with a covalent warhead for long-lasting inhibition
Author
Abstract
The synthesis and in vitro properties of six analogues of the selective glucocorticoid receptor (GR) agonist GSK866, bearing a warhead for covalent linkage to the glucocorticoid receptor, is described.
Language
English
Source (journal)
Bioorganic and medicinal chemistry letters. - Oxford
Publication
Oxford : 2016
ISSN
0960-894X
Volume/pages
26:20(2016), p. 5032-5038
ISI
000385498500036
Full text (Publisher's DOI)
Full text (open access)
Full text (publisher's version - intranet only)
UAntwerpen
Faculty/Department
Research group
Publication type
Subject
Affiliation
Publications with a UAntwerp address
External links
Web of Science
Record
Identification
Creation 22.09.2016
Last edited 08.06.2017
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